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Assay Detail

CHEMBL4732773

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ADMET
Cytotoxicity against human HaCaT cells after 24 hrs by MTT assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type ADMET
Organism Homo sapiens
Cell Type HaCaT
Confidence 1 — Organism
Curated By Autocuration

Target

HaCaT (CHEMBL614392)
Type CELL-LINE
Organism Homo sapiens

Publication

Sulfonium-based liposome-encapsulated antibiotics deliver a synergistic antibacterial activity
Patel, Anjali, Dey, Subhasis, Shokeen, Kamal, Karpinski, Tomasz M., Sivaprakasam, Senthilkumar, Kumar, Sachin, Manna, Debasis
RSC Med Chem (2021) 12 : 1005 -1015
PubMed 34223166 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 4.73 5.10

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1440 TETRACYCLINE 4.0 1 5.10
CHEMBL4751685 1 4.57
CHEMBL1082 AMOXICILLIN 4.0 1 4.53

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1440 TETRACYCLINE IC50 = 8000.0 nM 5.10
CHEMBL4751685 IC50 = 27000.0 nM 4.57
CHEMBL1082 AMOXICILLIN IC50 = 29410.0 nM 4.53