Assay Detail
Binding
CHEMBL4739810
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human GPR139 expressed in CHO-K1 cells assessed as induction of beta-arrestin 2 recruitment incubated for 90 mins by PathHunter assay
133
Total Activities
129
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | CHO-K1 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Probable G-protein coupled receptor 139 (CHEMBL3632455) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Gpr139 receptor modulators
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 133 | 8.65 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4742901 | — | — | 1 | 9.00 |
| CHEMBL4754576 | — | — | 1 | 9.00 |
| CHEMBL4764967 | — | — | 1 | 9.00 |
| CHEMBL4743662 | — | — | 1 | 9.00 |
| CHEMBL4754565 | — | — | 1 | 9.00 |
| CHEMBL4753388 | — | — | 1 | 9.00 |
| CHEMBL4746401 | — | — | 1 | 9.00 |
| CHEMBL4780358 | — | — | 1 | 9.00 |
| CHEMBL4750914 | — | — | 1 | 9.00 |
| CHEMBL4764290 | — | — | 1 | 9.00 |
| CHEMBL4800338 | — | — | 1 | 9.00 |
| CHEMBL4744927 | — | — | 1 | 9.00 |
| CHEMBL4762126 | — | — | 1 | 9.00 |
| CHEMBL4743612 | — | — | 1 | 9.00 |
| CHEMBL4789252 | — | — | 1 | 9.00 |
| CHEMBL4792732 | — | — | 1 | 9.00 |
| CHEMBL4757506 | — | — | 2 | 9.00 |
| CHEMBL4748306 | — | — | 1 | 9.00 |
| CHEMBL4759991 | — | — | 1 | 9.00 |
| CHEMBL4740491 | — | — | 1 | 9.00 |
| CHEMBL4782901 | — | — | 1 | 9.00 |
| CHEMBL4754735 | — | — | 1 | 9.00 |
| CHEMBL4756243 | — | — | 1 | 9.00 |
| CHEMBL4792896 | — | — | 1 | 9.00 |
| CHEMBL4748076 | — | — | 1 | 9.00 |
| CHEMBL4791193 | — | — | 1 | 9.00 |
| CHEMBL4756356 | — | — | 1 | 9.00 |
| CHEMBL4762651 | — | — | 1 | 9.00 |
| CHEMBL4765018 | — | — | 1 | 9.00 |
| CHEMBL4753640 | — | — | 1 | 9.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4750288 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4764967 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4791193 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4754576 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4742949 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4756356 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4799647 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4762651 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4786542 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4765018 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4753640 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4782901 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4790949 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4792732 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4798385 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4793093 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4752808 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4761154 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4751501 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4751304 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4756431 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4758841 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4753388 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4743662 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4740491 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4759991 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4748306 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4742901 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4789252 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4757506 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4743612 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4762126 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4754735 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4744927 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4754565 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4746401 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4780358 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4748076 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4750914 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4764290 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4800338 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4792896 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4756243 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL4754043 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL4747632 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL4799618 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL4764506 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL4758561 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL4750692 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL4798029 | — | EC50 | = | 10.0 | nM | 8.00 |