Assay Detail
Binding
CHEMBL4765713
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of TrkA (unknown origin)
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
High affinity nerve growth factor receptor (CHEMBL2815) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Indole-like Trk receptor antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 13 | 8.01 | 8.44 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL104519 | — | — | 1 | 8.44 |
| CHEMBL104333 | — | — | 1 | 8.42 |
| CHEMBL104279 | — | — | 1 | 8.38 |
| CHEMBL4788922 | — | — | 1 | 8.28 |
| CHEMBL106226 | — | — | 1 | 8.07 |
| CHEMBL4798255 | — | — | 1 | 8.04 |
| CHEMBL322153 | — | — | 1 | 8.00 |
| CHEMBL321955 | — | — | 1 | 7.95 |
| CHEMBL471375 | — | — | 1 | 7.59 |
| CHEMBL4074055 | — | — | 1 | 7.57 |
| CHEMBL476643 | — | — | 1 | 7.33 |
| CHEMBL382707 | — | — | 1 | - |
| CHEMBL261425 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL104519 | — | IC50 | = | 3.66 | nM | 8.44 |
| CHEMBL104333 | — | IC50 | = | 3.78 | nM | 8.42 |
| CHEMBL104279 | — | IC50 | = | 4.17 | nM | 8.38 |
| CHEMBL4788922 | — | IC50 | = | 5.22 | nM | 8.28 |
| CHEMBL106226 | — | IC50 | = | 8.49 | nM | 8.07 |
| CHEMBL4798255 | — | IC50 | = | 9.17 | nM | 8.04 |
| CHEMBL322153 | — | IC50 | = | 10.09 | nM | 8.00 |
| CHEMBL321955 | — | IC50 | = | 11.14 | nM | 7.95 |
| CHEMBL471375 | — | IC50 | = | 25.7 | nM | 7.59 |
| CHEMBL4074055 | — | IC50 | = | 27.21 | nM | 7.57 |
| CHEMBL476643 | — | IC50 | = | 46.34 | nM | 7.33 |
| CHEMBL382707 | — | IC50 | > | 10000.0 | nM | - |
| CHEMBL261425 | — | IC50 | > | 10000.0 | nM | - |