Assay Detail
Binding
CHEMBL4767577
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Inhibition of mouse GTA4 receptor
8
Total Activities
8
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Novel mouse GABA uptake inhibitors with enhanced inhibitory activity toward mGAT3/4 and their effect on pain threshold in mice.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 8 | 5.24 | 5.78 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4779064 | — | — | 1 | 5.78 |
| CHEMBL419823 | — | — | 1 | 5.71 |
| CHEMBL4566905 | — | — | 1 | 5.20 |
| CHEMBL3289575 | — | — | 1 | 5.04 |
| CHEMBL96 | GAMMA-AMINOBUTYRIC ACID | 1.0 | 1 | 4.48 |
| CHEMBL297569 | BETA-ALANINE | — | 1 | - |
| CHEMBL4793097 | — | — | 1 | - |
| CHEMBL4789121 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4779064 | — | IC50 | = | 1659.59 | nM | 5.78 |
| CHEMBL419823 | — | IC50 | = | 1949.84 | nM | 5.71 |
| CHEMBL4566905 | — | IC50 | = | 6309.57 | nM | 5.20 |
| CHEMBL3289575 | — | IC50 | = | 9120.11 | nM | 5.04 |
| CHEMBL96 | GAMMA-AMINOBUTYRIC ACID | IC50 | = | 33113.11 | nM | 4.48 |
| CHEMBL297569 | BETA-ALANINE | IC50 | = | 109647.82 | nM | - |
| CHEMBL4793097 | — | IC50 | = | 301995.17 | nM | - |
| CHEMBL4789121 | — | IC50 | = | 301995.17 | nM | - |