Assay Detail
Functional
CHEMBL4767683
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Antiproliferative activity against human U87MG cells assessed as cell growth inhibition measured after 72 hrs by SRB assay
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | U-87MG ATCC |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Efficient identification of novel anti-glioma lead compounds by machine learning models.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 19 | 4.97 | 5.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4061960 | — | — | 1 | 5.48 |
| CHEMBL4103684 | — | — | 1 | 5.41 |
| CHEMBL4070585 | — | — | 1 | 5.31 |
| CHEMBL4073310 | — | — | 1 | 5.28 |
| CHEMBL4100154 | — | — | 1 | 5.24 |
| CHEMBL4102608 | — | — | 1 | 5.17 |
| CHEMBL4072698 | — | — | 1 | 5.02 |
| CHEMBL4793298 | — | — | 1 | 5.01 |
| CHEMBL4092551 | — | — | 1 | 5.00 |
| CHEMBL4776452 | — | — | 1 | 4.98 |
| CHEMBL4799550 | — | — | 1 | 4.91 |
| CHEMBL1269013 | — | — | 1 | 4.90 |
| CHEMBL2029363 | — | — | 1 | 4.87 |
| CHEMBL4068974 | — | — | 1 | 4.87 |
| CHEMBL4778320 | — | — | 1 | 4.72 |
| CHEMBL4079425 | — | — | 1 | 4.49 |
| CHEMBL4059707 | — | — | 1 | 4.45 |
| CHEMBL4093415 | — | — | 1 | 4.35 |
| CHEMBL810 | TEMOZOLOMIDE | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4061960 | — | EC50 | = | 3300.0 | nM | 5.48 |
| CHEMBL4103684 | — | EC50 | = | 3900.0 | nM | 5.41 |
| CHEMBL4070585 | — | EC50 | = | 4900.0 | nM | 5.31 |
| CHEMBL4073310 | — | EC50 | = | 5200.0 | nM | 5.28 |
| CHEMBL4100154 | — | EC50 | = | 5800.0 | nM | 5.24 |
| CHEMBL4102608 | — | EC50 | = | 6800.0 | nM | 5.17 |
| CHEMBL4072698 | — | EC50 | = | 9500.0 | nM | 5.02 |
| CHEMBL4793298 | — | EC50 | = | 9800.0 | nM | 5.01 |
| CHEMBL4092551 | — | EC50 | = | 10100.0 | nM | 5.00 |
| CHEMBL4776452 | — | EC50 | = | 10500.0 | nM | 4.98 |
| CHEMBL4799550 | — | EC50 | = | 12300.0 | nM | 4.91 |
| CHEMBL1269013 | — | EC50 | = | 12600.0 | nM | 4.90 |
| CHEMBL2029363 | — | EC50 | = | 13400.0 | nM | 4.87 |
| CHEMBL4068974 | — | EC50 | = | 13400.0 | nM | 4.87 |
| CHEMBL4778320 | — | EC50 | = | 19200.0 | nM | 4.72 |
| CHEMBL4079425 | — | EC50 | = | 32300.0 | nM | 4.49 |
| CHEMBL4059707 | — | EC50 | = | 35400.0 | nM | 4.45 |
| CHEMBL4093415 | — | EC50 | = | 45100.0 | nM | 4.35 |
| CHEMBL810 | TEMOZOLOMIDE | EC50 | > | 200000.0 | nM | - |