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Assay Detail

CHEMBL4774476

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antigiardial activity against Giardia intestinalis WB ATCC 30957 incubated for 72 hrs by hemocytometric counting method
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Giardia intestinalis
Confidence 1 — Organism
Curated By Autocuration

Target

Giardia intestinalis (CHEMBL612652)
Type ORGANISM
Organism Giardia intestinalis

Publication

Anti-Giardia Drug Discovery: Current Status and Gut Feelings.
Riches A,Hart CJS,Trenholme KR,Skinner-Adams TS
J Med Chem (2020) 63 : 13330 -13354
PubMed 32869995 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 3 5.63 6.01

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4795316 1 6.01
CHEMBL4786380 1 5.25
CHEMBL4787668 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4795316 IC50 = 970.0 nM 6.01
CHEMBL4786380 IC50 = 5600.0 nM 5.25
CHEMBL4787668 IC50 = 144800.0 nM -