Assay Detail
Binding
CHEMBL4806265
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of casein kinase 1delta (unknown origin)
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Small molecule inhibitors of cdk12/cdk13
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 11 | 6.08 | 8.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4855324 | — | — | 1 | 8.40 |
| CHEMBL4849960 | — | — | 1 | 6.48 |
| CHEMBL4856935 | — | — | 1 | 6.40 |
| CHEMBL4849684 | — | — | 1 | 6.38 |
| CHEMBL4868958 | — | — | 1 | 6.06 |
| CHEMBL4867928 | — | — | 1 | 5.90 |
| CHEMBL4877117 | — | — | 1 | 5.53 |
| CHEMBL4847754 | — | — | 1 | 5.32 |
| CHEMBL4868638 | — | — | 1 | 5.22 |
| CHEMBL4852083 | — | — | 1 | 5.07 |
| CHEMBL4856716 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4855324 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4849960 | — | IC50 | = | 333.0 | nM | 6.48 |
| CHEMBL4856935 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL4849684 | — | IC50 | = | 419.0 | nM | 6.38 |
| CHEMBL4868958 | — | IC50 | = | 870.0 | nM | 6.06 |
| CHEMBL4867928 | — | IC50 | = | 1257.0 | nM | 5.90 |
| CHEMBL4877117 | — | IC50 | = | 2935.0 | nM | 5.53 |
| CHEMBL4847754 | — | IC50 | = | 4745.0 | nM | 5.32 |
| CHEMBL4868638 | — | IC50 | = | 6065.0 | nM | 5.22 |
| CHEMBL4852083 | — | IC50 | = | 8600.0 | nM | 5.07 |
| CHEMBL4856716 | — | IC50 | > | 9900.0 | nM | - |