Assay Detail
Binding
CHEMBL4808052
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Inhibition of HIPK4 (unknown origin)
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Homeodomain-interacting protein kinase 4 (CHEMBL1075167) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Hipk inhibitors and methods of use thereof
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 10 | 8.03 | 8.55 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4855209 | — | — | 1 | 8.55 |
| CHEMBL1336 | SORAFENIB | 4.0 | 1 | 8.52 |
| CHEMBL4859179 | — | — | 1 | 8.48 |
| CHEMBL4850066 | — | — | 1 | 8.29 |
| CHEMBL4855979 | — | — | 1 | 8.28 |
| CHEMBL4870763 | — | — | 1 | 8.02 |
| CHEMBL4874174 | — | — | 1 | 7.72 |
| CHEMBL4847460 | — | — | 1 | 7.64 |
| CHEMBL4875968 | — | — | 1 | 7.50 |
| CHEMBL4853006 | — | — | 1 | 7.31 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4855209 | — | IC50 | = | 2.8 | nM | 8.55 |
| CHEMBL1336 | SORAFENIB | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL4859179 | — | IC50 | = | 3.3 | nM | 8.48 |
| CHEMBL4850066 | — | IC50 | = | 5.1 | nM | 8.29 |
| CHEMBL4855979 | — | IC50 | = | 5.2 | nM | 8.28 |
| CHEMBL4870763 | — | IC50 | = | 9.6 | nM | 8.02 |
| CHEMBL4874174 | — | IC50 | = | 19.0 | nM | 7.72 |
| CHEMBL4847460 | — | IC50 | = | 23.0 | nM | 7.64 |
| CHEMBL4875968 | — | IC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4853006 | — | IC50 | = | 49.0 | nM | 7.31 |