Assay Detail
Functional
CHEMBL4811327
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antischistosomal activity against Schistosoma mansoni Liberian NTS incubated for 72 hrs by microscopic method
26
Total Activities
26
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Schistosoma mansoni |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Chemotherapy for human schistosomiasis: how far have we come? What's new? Where do we go from here?
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 26 | 5.82 | 6.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2313136 | — | — | 1 | 6.70 |
| CHEMBL3637921 | — | — | 1 | 6.40 |
| CHEMBL3637922 | — | — | 1 | 6.40 |
| CHEMBL607707 | PELITINIB | 2.0 | 1 | 6.30 |
| CHEMBL534797 | — | — | 1 | 6.22 |
| CHEMBL4855202 | — | — | 1 | 6.22 |
| CHEMBL91867 | — | — | 1 | 6.16 |
| CHEMBL3637864 | — | — | 1 | 6.10 |
| CHEMBL3637865 | — | — | 1 | 6.10 |
| CHEMBL1367316 | — | — | 1 | 6.05 |
| CHEMBL228814 | ISPINESIB | 2.0 | 1 | 6.05 |
| CHEMBL15928 | GR-127935 | — | 1 | 5.92 |
| CHEMBL88272 | — | — | 1 | 5.82 |
| CHEMBL16687 | CGS-15943 | — | 1 | 5.77 |
| CHEMBL531611 | — | — | 1 | 5.75 |
| CHEMBL59030 | — | — | 1 | 5.68 |
| CHEMBL3637915 | — | — | 1 | 5.66 |
| CHEMBL545853 | — | — | 1 | 5.58 |
| CHEMBL598279 | — | — | 1 | 5.57 |
| CHEMBL565436 | — | — | 1 | 5.54 |
| CHEMBL537152 | — | — | 1 | 5.47 |
| CHEMBL3545403 | BMS-833923 | 2.0 | 1 | 5.46 |
| CHEMBL10835 | — | — | 1 | 5.33 |
| CHEMBL513909 | BI-2536 | 2.0 | 1 | 5.20 |
| CHEMBL238125 | — | — | 1 | 5.14 |
| CHEMBL4850244 | — | — | 1 | 4.78 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2313136 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL3637921 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL3637922 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL607707 | PELITINIB | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL534797 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL4855202 | — | IC50 | = | 600.0 | nM | 6.22 |
| CHEMBL91867 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL3637864 | — | IC50 | = | 800.0 | nM | 6.10 |
| CHEMBL3637865 | — | IC50 | = | 800.0 | nM | 6.10 |
| CHEMBL1367316 | — | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL228814 | ISPINESIB | IC50 | = | 900.0 | nM | 6.05 |
| CHEMBL15928 | GR-127935 | IC50 | = | 1200.0 | nM | 5.92 |
| CHEMBL88272 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL16687 | CGS-15943 | IC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL531611 | — | IC50 | = | 1800.0 | nM | 5.75 |
| CHEMBL59030 | — | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL3637915 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL545853 | — | IC50 | = | 2600.0 | nM | 5.58 |
| CHEMBL598279 | — | IC50 | = | 2700.0 | nM | 5.57 |
| CHEMBL565436 | — | IC50 | = | 2900.0 | nM | 5.54 |
| CHEMBL537152 | — | IC50 | = | 3400.0 | nM | 5.47 |
| CHEMBL3545403 | BMS-833923 | IC50 | = | 3500.0 | nM | 5.46 |
| CHEMBL10835 | — | IC50 | = | 4700.0 | nM | 5.33 |
| CHEMBL513909 | BI-2536 | IC50 | = | 6300.0 | nM | 5.20 |
| CHEMBL238125 | — | IC50 | = | 7200.0 | nM | 5.14 |
| CHEMBL4850244 | — | IC50 | = | 16700.0 | nM | 4.78 |