Assay Detail
Binding
CHEMBL4814673
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Inhibition of porcine pancreatic alpha-amylase using 1% starch as substrate preincubated for 10 mins followed by substrate addition and measured after 10 mins by absorbance method
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Sus scrofa |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Metronidazole-conjugates: A comprehensive review of recent developments towards synthesis and medicinal perspective.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 21 | 5.99 | 6.42 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4861741 | — | — | 1 | 6.42 |
| CHEMBL4864128 | — | — | 1 | 5.78 |
| CHEMBL404271 | ACARBOSE | 4.0 | 1 | 5.78 |
| CHEMBL188521 | — | — | 1 | - |
| CHEMBL4854163 | — | — | 1 | - |
| CHEMBL4851123 | — | — | 1 | - |
| CHEMBL4846195 | — | — | 1 | - |
| CHEMBL4865236 | — | — | 1 | - |
| CHEMBL4866987 | — | — | 1 | - |
| CHEMBL4875625 | — | — | 1 | - |
| CHEMBL4868815 | — | — | 1 | - |
| CHEMBL4860734 | — | — | 1 | - |
| CHEMBL4869717 | — | — | 1 | - |
| CHEMBL4876409 | — | — | 1 | - |
| CHEMBL4876278 | — | — | 1 | - |
| CHEMBL4859800 | — | — | 1 | - |
| CHEMBL4859605 | — | — | 1 | - |
| CHEMBL4867711 | — | — | 1 | - |
| CHEMBL4866166 | — | — | 1 | - |
| CHEMBL4866437 | — | — | 1 | - |
| CHEMBL4871075 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4861741 | — | IC50 | = | 380.0 | nM | 6.42 |
| CHEMBL4864128 | — | IC50 | = | 1660.0 | nM | 5.78 |
| CHEMBL404271 | ACARBOSE | IC50 | = | 1660.0 | nM | 5.78 |
| CHEMBL188521 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4854163 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4851123 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4846195 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4865236 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4866987 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4875625 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4868815 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4860734 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4869717 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4876409 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4876278 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4859800 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4859605 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4867711 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4866166 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4866437 | — | IC50 | < | 2980.0 | nM | - |
| CHEMBL4871075 | — | IC50 | < | 2980.0 | nM | - |