Assay Detail
Functional
CHEMBL4819529
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Agonist activity at beta2 adrenoceptor (unknown origin)
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Recent Advances in β<sub>2</sub>-Agonists for Treatment of Chronic Respiratory Diseases and Heart Failure.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 4 | 8.76 | 10.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL605846 | OLODATEROL | 4.0 | 1 | 10.70 |
| CHEMBL1095777 | INDACATEROL | 4.0 | 1 | 9.10 |
| CHEMBL4874511 | — | — | 1 | 7.66 |
| CHEMBL1615159 | — | — | 1 | 7.57 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL605846 | OLODATEROL | EC50 | = | 0.02 | nM | 10.70 |
| CHEMBL1095777 | INDACATEROL | EC50 | = | 0.79 | nM | 9.10 |
| CHEMBL4874511 | — | EC50 | = | 21.8 | nM | 7.66 |
| CHEMBL1615159 | — | EC50 | = | 27.0 | nM | 7.57 |