Assay Detail
ADMET
CHEMBL4824671
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Cytotoxicity against human glomerular mesangial cells incubated for 12 hrs by MTT assay
25
Total Activities
25
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | ADMET |
| Organism | Homo sapiens |
| Cell Type | Glomerular mesangial cell |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Novel Broad-Spectrum Antimicrobial Peptide Derived from Anoplin and Its Activity on Bacterial Pneumonia in Mice.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 25 | 4.46 | 5.83 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL412927 | MELITTIN | — | 1 | 5.83 |
| CHEMBL4860493 | — | — | 1 | 4.95 |
| CHEMBL4850509 | — | — | 1 | 4.70 |
| CHEMBL4862426 | — | — | 1 | 4.60 |
| CHEMBL4853738 | — | — | 1 | 4.41 |
| CHEMBL4871749 | — | — | 1 | 4.39 |
| CHEMBL4874973 | — | — | 1 | 4.32 |
| CHEMBL4859995 | — | — | 1 | 4.30 |
| CHEMBL4870321 | — | — | 1 | 4.28 |
| CHEMBL4871296 | — | — | 1 | 4.10 |
| CHEMBL4865196 | — | — | 1 | 4.05 |
| CHEMBL4855065 | — | — | 1 | 4.04 |
| CHEMBL4845719 | — | — | 1 | 4.01 |
| CHEMBL4865224 | — | — | 1 | - |
| CHEMBL2397513 | — | — | 1 | - |
| CHEMBL4850027 | — | — | 1 | - |
| CHEMBL2396875 | ANOPLIN | — | 1 | - |
| CHEMBL4852506 | — | — | 1 | - |
| CHEMBL4845856 | — | — | 1 | - |
| CHEMBL4862255 | — | — | 1 | - |
| CHEMBL4877165 | — | — | 1 | - |
| CHEMBL4877580 | — | — | 1 | - |
| CHEMBL4858900 | — | — | 1 | - |
| CHEMBL4859713 | — | — | 1 | - |
| CHEMBL4854087 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL412927 | MELITTIN | IC50 | = | 1490.0 | nM | 5.83 |
| CHEMBL4860493 | — | IC50 | = | 11240.0 | nM | 4.95 |
| CHEMBL4850509 | — | IC50 | = | 19770.0 | nM | 4.70 |
| CHEMBL4862426 | — | IC50 | = | 25170.0 | nM | 4.60 |
| CHEMBL4853738 | — | IC50 | = | 38970.0 | nM | 4.41 |
| CHEMBL4871749 | — | IC50 | = | 40250.0 | nM | 4.39 |
| CHEMBL4874973 | — | IC50 | = | 48210.0 | nM | 4.32 |
| CHEMBL4859995 | — | IC50 | = | 49490.0 | nM | 4.30 |
| CHEMBL4870321 | — | IC50 | = | 52620.0 | nM | 4.28 |
| CHEMBL4871296 | — | IC50 | = | 80210.0 | nM | 4.10 |
| CHEMBL4865196 | — | IC50 | = | 88890.0 | nM | 4.05 |
| CHEMBL4855065 | — | IC50 | = | 91880.0 | nM | 4.04 |
| CHEMBL4845719 | — | IC50 | = | 98280.0 | nM | 4.01 |
| CHEMBL4865224 | — | IC50 | = | 104530.0 | nM | - |
| CHEMBL2397513 | — | IC50 | >= | 512000.0 | nM | - |
| CHEMBL4850027 | — | IC50 | >= | 512000.0 | nM | - |
| CHEMBL2396875 | ANOPLIN | IC50 | >= | 512000.0 | nM | - |
| CHEMBL4852506 | — | IC50 | >= | 512000.0 | nM | - |
| CHEMBL4845856 | — | IC50 | = | 209210.0 | nM | - |
| CHEMBL4862255 | — | IC50 | >= | 512000.0 | nM | - |
| CHEMBL4877165 | — | IC50 | >= | 512000.0 | nM | - |
| CHEMBL4877580 | — | IC50 | >= | 512000.0 | nM | - |
| CHEMBL4858900 | — | IC50 | >= | 512000.0 | nM | - |
| CHEMBL4859713 | — | IC50 | >= | 512000.0 | nM | - |
| CHEMBL4854087 | — | IC50 | >= | 512000.0 | nM | - |