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Assay Detail

CHEMBL4825922

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Functional
Antiviral activity against Respiratory syncytial virus A2 infected in human Hep2 cells by Plaque reduction assay
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human respiratory syncytial virus
Cell Type HEp-2
Confidence 1 — Organism
Curated By Autocuration

Target

Human orthopneumovirus (CHEMBL613127)
Type ORGANISM
Organism Human orthopneumovirus

Publication

Discovery of Sisunatovir (RV521), an Inhibitor of Respiratory Syncytial Virus Fusion.
Cockerill GS, Angell RM, Bedernjak A, Chuckowree I, Fraser I, Gascon-Simorte J, Gilman MSA, Good JAD, Harland R, Johnson SM, Ludes-Meyers JH, Littler E, Lumley J, Lunn G, Mathews N, McLellan JS, Paradowski M, Peeples ME, Scott C, Tait D, Taylor G, Thom M, Thomas E, Villalonga Barber C, Ward SE, Watterson D, Williams G, Young P, Powell K.
J Med Chem (2021) 64 : 3658 -3676
PubMed 33729773 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 4 7.95 9.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4855358 1 9.30
CHEMBL4847062 1 7.86
CHEMBL4866951 1 7.68
CHEMBL4871056 1 6.97

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4855358 EC50 = 0.5 nM 9.30
CHEMBL4847062 EC50 = 13.7 nM 7.86
CHEMBL4866951 EC50 = 21.1 nM 7.68
CHEMBL4871056 EC50 = 106.7 nM 6.97