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Assay Detail

CHEMBL4837569

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to GABBA alpha5 (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Gamma-aminobutyric acid receptor subunit alpha-5 (CHEMBL5112)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Pharmacological Analysis of the Anti-inflammatory and Antiallodynic Effects of Zinagrandinolide E from <i>Zinnia grandiflora</i> in Mice.
Reyes-Pérez VI, Granados-Soto V, Rangel-Grimaldo M, Déciga-Campos M, Mata R.
J Nat Prod (2021) 84 : 713 -723
PubMed 32870011 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 9.20 9.20

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL407 FLUMAZENIL 4.0 1 9.20

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL407 FLUMAZENIL Ki = 0.631 nM 9.20