Assay Detail
Binding
CHEMBL4838702
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of MERTK (unknown origin)
35
Total Activities
35
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
UNC5293, a potent, orally available and highly MERTK-selective inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 35 | 8.44 | 9.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4877347 | — | — | 1 | 9.05 |
| CHEMBL4857351 | — | — | 1 | 9.05 |
| CHEMBL4866538 | — | — | 1 | 8.92 |
| CHEMBL4862333 | — | — | 1 | 8.92 |
| CHEMBL4867544 | — | — | 1 | 8.89 |
| CHEMBL4856976 | — | — | 1 | 8.82 |
| CHEMBL4847691 | — | — | 1 | 8.80 |
| CHEMBL4851097 | — | — | 1 | 8.72 |
| CHEMBL4877792 | — | — | 1 | 8.64 |
| CHEMBL4857561 | — | — | 1 | 8.64 |
| CHEMBL4878347 | — | — | 1 | 8.62 |
| CHEMBL4850498 | — | — | 1 | 8.59 |
| CHEMBL4847256 | — | — | 1 | 8.55 |
| CHEMBL4875352 | — | — | 1 | 8.52 |
| CHEMBL4849169 | — | — | 1 | 8.52 |
| CHEMBL4877058 | — | — | 1 | 8.51 |
| CHEMBL4854055 | — | — | 1 | 8.47 |
| CHEMBL4878774 | — | — | 1 | 8.40 |
| CHEMBL4862062 | — | — | 1 | 8.38 |
| CHEMBL4868941 | — | — | 1 | 8.36 |
| CHEMBL4875531 | — | — | 1 | 8.35 |
| CHEMBL4853524 | — | — | 1 | 8.34 |
| CHEMBL4878118 | — | — | 1 | 8.32 |
| CHEMBL4854618 | — | — | 1 | 8.30 |
| CHEMBL4851303 | — | — | 1 | 8.28 |
| CHEMBL4873478 | — | — | 1 | 8.26 |
| CHEMBL4846907 | — | — | 1 | 8.21 |
| CHEMBL4861169 | — | — | 1 | 8.21 |
| CHEMBL4845859 | — | — | 1 | 8.19 |
| CHEMBL4848248 | — | — | 1 | 8.14 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4877347 | — | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL4857351 | — | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL4866538 | — | IC50 | = | 1.2 | nM | 8.92 |
| CHEMBL4862333 | — | IC50 | = | 1.2 | nM | 8.92 |
| CHEMBL4867544 | — | IC50 | = | 1.3 | nM | 8.89 |
| CHEMBL4856976 | — | IC50 | = | 1.5 | nM | 8.82 |
| CHEMBL4847691 | — | IC50 | = | 1.6 | nM | 8.80 |
| CHEMBL4851097 | — | IC50 | = | 1.9 | nM | 8.72 |
| CHEMBL4877792 | — | IC50 | = | 2.3 | nM | 8.64 |
| CHEMBL4857561 | — | IC50 | = | 2.3 | nM | 8.64 |
| CHEMBL4878347 | — | IC50 | = | 2.4 | nM | 8.62 |
| CHEMBL4850498 | — | IC50 | = | 2.6 | nM | 8.59 |
| CHEMBL4847256 | — | IC50 | = | 2.8 | nM | 8.55 |
| CHEMBL4875352 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL4849169 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL4877058 | — | IC50 | = | 3.1 | nM | 8.51 |
| CHEMBL4854055 | — | IC50 | = | 3.4 | nM | 8.47 |
| CHEMBL4878774 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL4862062 | — | IC50 | = | 4.2 | nM | 8.38 |
| CHEMBL4868941 | — | IC50 | = | 4.4 | nM | 8.36 |
| CHEMBL4875531 | — | IC50 | = | 4.5 | nM | 8.35 |
| CHEMBL4853524 | — | IC50 | = | 4.6 | nM | 8.34 |
| CHEMBL4878118 | — | IC50 | = | 4.8 | nM | 8.32 |
| CHEMBL4854618 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL4851303 | — | IC50 | = | 5.2 | nM | 8.28 |
| CHEMBL4873478 | — | IC50 | = | 5.5 | nM | 8.26 |
| CHEMBL4846907 | — | IC50 | = | 6.2 | nM | 8.21 |
| CHEMBL4861169 | — | IC50 | = | 6.1 | nM | 8.21 |
| CHEMBL4845859 | — | IC50 | = | 6.5 | nM | 8.19 |
| CHEMBL4848248 | — | IC50 | = | 7.2 | nM | 8.14 |
| CHEMBL4854016 | — | IC50 | = | 7.9 | nM | 8.10 |
| CHEMBL4866585 | — | IC50 | = | 8.5 | nM | 8.07 |
| CHEMBL4861342 | — | IC50 | = | 9.5 | nM | 8.02 |
| CHEMBL4855700 | — | IC50 | = | 13.0 | nM | 7.89 |
| CHEMBL4862025 | — | IC50 | = | 30.0 | nM | 7.52 |