Assay Detail
Binding
CHEMBL4838705
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Inhibition of FLT3 (unknown origin)
35
Total Activities
35
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Receptor-type tyrosine-protein kinase FLT3 (CHEMBL1974) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
UNC5293, a potent, orally available and highly MERTK-selective inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 35 | 6.33 | 8.18 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4866538 | — | — | 1 | 8.18 |
| CHEMBL4857351 | — | — | 1 | 7.68 |
| CHEMBL4856976 | — | — | 1 | 7.26 |
| CHEMBL4877347 | — | — | 1 | 7.05 |
| CHEMBL4862333 | — | — | 1 | 6.92 |
| CHEMBL4867544 | — | — | 1 | 6.82 |
| CHEMBL4878774 | — | — | 1 | 6.70 |
| CHEMBL4851097 | — | — | 1 | 6.68 |
| CHEMBL4861169 | — | — | 1 | 6.68 |
| CHEMBL4847691 | — | — | 1 | 6.66 |
| CHEMBL4849169 | — | — | 1 | 6.55 |
| CHEMBL4854618 | — | — | 1 | 6.54 |
| CHEMBL4854055 | — | — | 1 | 6.46 |
| CHEMBL4877792 | — | — | 1 | 6.43 |
| CHEMBL4875352 | — | — | 1 | 6.40 |
| CHEMBL4878347 | — | — | 1 | 6.39 |
| CHEMBL4878118 | — | — | 1 | 6.38 |
| CHEMBL4877058 | — | — | 1 | 6.31 |
| CHEMBL4857561 | — | — | 1 | 6.28 |
| CHEMBL4861342 | — | — | 1 | 6.24 |
| CHEMBL4873478 | — | — | 1 | 6.23 |
| CHEMBL4847256 | — | — | 1 | 6.21 |
| CHEMBL4850498 | — | — | 1 | 6.17 |
| CHEMBL4862062 | — | — | 1 | 6.08 |
| CHEMBL4848248 | — | — | 1 | 6.07 |
| CHEMBL4851303 | — | — | 1 | 5.96 |
| CHEMBL4846907 | — | — | 1 | 5.96 |
| CHEMBL4868941 | — | — | 1 | 5.89 |
| CHEMBL4845859 | — | — | 1 | 5.82 |
| CHEMBL4866585 | — | — | 1 | 5.78 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4866538 | — | IC50 | = | 6.6 | nM | 8.18 |
| CHEMBL4857351 | — | IC50 | = | 21.0 | nM | 7.68 |
| CHEMBL4856976 | — | IC50 | = | 55.0 | nM | 7.26 |
| CHEMBL4877347 | — | IC50 | = | 90.0 | nM | 7.05 |
| CHEMBL4862333 | — | IC50 | = | 120.0 | nM | 6.92 |
| CHEMBL4867544 | — | IC50 | = | 150.0 | nM | 6.82 |
| CHEMBL4878774 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL4851097 | — | IC50 | = | 210.0 | nM | 6.68 |
| CHEMBL4861169 | — | IC50 | = | 210.0 | nM | 6.68 |
| CHEMBL4847691 | — | IC50 | = | 220.0 | nM | 6.66 |
| CHEMBL4849169 | — | IC50 | = | 280.0 | nM | 6.55 |
| CHEMBL4854618 | — | IC50 | = | 290.0 | nM | 6.54 |
| CHEMBL4854055 | — | IC50 | = | 350.0 | nM | 6.46 |
| CHEMBL4877792 | — | IC50 | = | 370.0 | nM | 6.43 |
| CHEMBL4875352 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL4878347 | — | IC50 | = | 410.0 | nM | 6.39 |
| CHEMBL4878118 | — | IC50 | = | 420.0 | nM | 6.38 |
| CHEMBL4877058 | — | IC50 | = | 490.0 | nM | 6.31 |
| CHEMBL4857561 | — | IC50 | = | 520.0 | nM | 6.28 |
| CHEMBL4861342 | — | IC50 | = | 580.0 | nM | 6.24 |
| CHEMBL4873478 | — | IC50 | = | 590.0 | nM | 6.23 |
| CHEMBL4847256 | — | IC50 | = | 620.0 | nM | 6.21 |
| CHEMBL4850498 | — | IC50 | = | 680.0 | nM | 6.17 |
| CHEMBL4862062 | — | IC50 | = | 840.0 | nM | 6.08 |
| CHEMBL4848248 | — | IC50 | = | 860.0 | nM | 6.07 |
| CHEMBL4846907 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL4851303 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL4868941 | — | IC50 | = | 1300.0 | nM | 5.89 |
| CHEMBL4845859 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL4866585 | — | IC50 | = | 1680.0 | nM | 5.78 |
| CHEMBL4853524 | — | IC50 | = | 1650.0 | nM | 5.78 |
| CHEMBL4854016 | — | IC50 | = | 1690.0 | nM | 5.77 |
| CHEMBL4875531 | — | IC50 | = | 4920.0 | nM | 5.31 |
| CHEMBL4862025 | — | IC50 | = | 7890.0 | nM | 5.10 |
| CHEMBL4855700 | — | IC50 | = | 10970.0 | nM | 4.96 |