Assay Detail
Binding
CHEMBL4843202
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Agonist activity at rat AMY3R (CT+RAMP3) expressed in tk-ts13 cells assessed as increase in intracellular cAMP level incuabted for 25 mins by CRE luciferase reporter gene assay
29
Total Activities
29
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Cell Type | tk-ts13 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Development of Cagrilintide, a Long-Acting Amylin Analogue.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 29 | 9.67 | 10.20 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4853852 | — | — | 1 | 10.20 |
| CHEMBL4857768 | — | — | 1 | 10.09 |
| CHEMBL4859695 | — | — | 1 | 10.08 |
| CHEMBL4860327 | — | — | 1 | 9.92 |
| CHEMBL4865624 | — | — | 1 | 9.89 |
| CHEMBL4866960 | — | — | 1 | 9.88 |
| CHEMBL4847769 | — | — | 1 | 9.85 |
| CHEMBL4859757 | — | — | 1 | 9.83 |
| CHEMBL4877066 | — | — | 1 | 9.80 |
| CHEMBL4872163 | — | — | 1 | 9.73 |
| CHEMBL4860505 | — | — | 1 | 9.63 |
| CHEMBL4847968 | — | — | 1 | 9.61 |
| CHEMBL4852769 | — | — | 1 | 9.58 |
| CHEMBL4873689 | — | — | 1 | 9.56 |
| CHEMBL4874471 | — | — | 1 | 9.56 |
| CHEMBL4863815 | — | — | 1 | 9.49 |
| CHEMBL4868506 | — | — | 1 | 9.47 |
| CHEMBL4860423 | — | — | 1 | 9.46 |
| CHEMBL4856338 | — | — | 1 | 9.31 |
| CHEMBL4854371 | — | — | 1 | 9.21 |
| CHEMBL4861227 | — | — | 1 | 8.99 |
| CHEMBL3989767 | CALCITONIN SALMON | 4.0 | 1 | - |
| CHEMBL2103758 | PRAMLINTIDE | 4.0 | 1 | - |
| CHEMBL4863501 | — | — | 1 | - |
| CHEMBL4856671 | — | — | 1 | - |
| CHEMBL4863929 | — | — | 1 | - |
| CHEMBL4853250 | — | — | 1 | - |
| CHEMBL4855949 | — | — | 1 | - |
| CHEMBL4846668 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4853852 | — | EC50 | = | 0.063 | nM | 10.20 |
| CHEMBL4857768 | — | EC50 | = | 0.082 | nM | 10.09 |
| CHEMBL4859695 | — | EC50 | = | 0.083 | nM | 10.08 |
| CHEMBL4860327 | — | EC50 | = | 0.121 | nM | 9.92 |
| CHEMBL4865624 | — | EC50 | = | 0.13 | nM | 9.89 |
| CHEMBL4866960 | — | EC50 | = | 0.132 | nM | 9.88 |
| CHEMBL4847769 | — | EC50 | = | 0.143 | nM | 9.85 |
| CHEMBL4859757 | — | EC50 | = | 0.147 | nM | 9.83 |
| CHEMBL4877066 | — | EC50 | = | 0.158 | nM | 9.80 |
| CHEMBL4872163 | — | EC50 | = | 0.188 | nM | 9.73 |
| CHEMBL4860505 | — | EC50 | = | 0.233 | nM | 9.63 |
| CHEMBL4847968 | — | EC50 | = | 0.246 | nM | 9.61 |
| CHEMBL4852769 | — | EC50 | = | 0.261 | nM | 9.58 |
| CHEMBL4873689 | — | EC50 | = | 0.278 | nM | 9.56 |
| CHEMBL4874471 | — | EC50 | = | 0.277 | nM | 9.56 |
| CHEMBL4863815 | — | EC50 | = | 0.321 | nM | 9.49 |
| CHEMBL4868506 | — | EC50 | = | 0.335 | nM | 9.47 |
| CHEMBL4860423 | — | EC50 | = | 0.348 | nM | 9.46 |
| CHEMBL4856338 | — | EC50 | = | 0.49 | nM | 9.31 |
| CHEMBL4854371 | — | EC50 | = | 0.623 | nM | 9.21 |
| CHEMBL4861227 | — | EC50 | = | 1.031 | nM | 8.99 |
| CHEMBL3989767 | CALCITONIN SALMON | EC50 | = | 0.001 | nM | - |
| CHEMBL2103758 | PRAMLINTIDE | EC50 | = | 0.004 | nM | - |
| CHEMBL4863501 | — | EC50 | - | — | - | |
| CHEMBL4856671 | — | EC50 | - | — | - | |
| CHEMBL4863929 | — | EC50 | - | — | - | |
| CHEMBL4853250 | — | EC50 | - | — | - | |
| CHEMBL4855949 | — | EC50 | - | — | - | |
| CHEMBL4846668 | — | EC50 | - | — | - |