Assay Detail
Binding
CHEMBL4843205
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Displacement of [125I]-amylin from human AMY3R (CTR+RAMP3) expressed in BHK-13 cells measured after 120 mins by scintillation proximity assay
19
Total Activities
19
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | BHK-13 |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Development of Cagrilintide, a Long-Acting Amylin Analogue.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 19 | 9.49 | 10.28 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4866960 | — | — | 1 | 10.28 |
| CHEMBL3989767 | CALCITONIN SALMON | 4.0 | 1 | 10.05 |
| CHEMBL2103758 | PRAMLINTIDE | 4.0 | 1 | 9.94 |
| CHEMBL4853852 | — | — | 1 | 9.86 |
| CHEMBL4860423 | — | — | 1 | 9.77 |
| CHEMBL4877066 | — | — | 1 | 9.73 |
| CHEMBL4872163 | — | — | 1 | 9.72 |
| CHEMBL4865624 | — | — | 1 | 9.67 |
| CHEMBL4868506 | — | — | 1 | 9.67 |
| CHEMBL4860327 | — | — | 1 | 9.53 |
| CHEMBL4863501 | — | — | 1 | 9.46 |
| CHEMBL4859757 | — | — | 1 | 9.45 |
| CHEMBL4853250 | — | — | 1 | 9.30 |
| CHEMBL4859695 | — | — | 1 | 9.14 |
| CHEMBL4855949 | — | — | 1 | 9.09 |
| CHEMBL4847968 | — | — | 1 | 8.97 |
| CHEMBL4863815 | — | — | 1 | 8.96 |
| CHEMBL4861227 | — | — | 1 | 8.89 |
| CHEMBL4863929 | — | — | 1 | 8.87 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4866960 | — | IC50 | = | 0.052 | nM | 10.28 |
| CHEMBL3989767 | CALCITONIN SALMON | IC50 | = | 0.089 | nM | 10.05 |
| CHEMBL2103758 | PRAMLINTIDE | IC50 | = | 0.114 | nM | 9.94 |
| CHEMBL4853852 | — | IC50 | = | 0.137 | nM | 9.86 |
| CHEMBL4860423 | — | IC50 | = | 0.17 | nM | 9.77 |
| CHEMBL4877066 | — | IC50 | = | 0.186 | nM | 9.73 |
| CHEMBL4872163 | — | IC50 | = | 0.192 | nM | 9.72 |
| CHEMBL4865624 | — | IC50 | = | 0.213 | nM | 9.67 |
| CHEMBL4868506 | — | IC50 | = | 0.216 | nM | 9.67 |
| CHEMBL4860327 | — | IC50 | = | 0.293 | nM | 9.53 |
| CHEMBL4863501 | — | IC50 | = | 0.35 | nM | 9.46 |
| CHEMBL4859757 | — | IC50 | = | 0.359 | nM | 9.45 |
| CHEMBL4853250 | — | IC50 | = | 0.499 | nM | 9.30 |
| CHEMBL4859695 | — | IC50 | = | 0.723 | nM | 9.14 |
| CHEMBL4855949 | — | IC50 | = | 0.818 | nM | 9.09 |
| CHEMBL4847968 | — | IC50 | = | 1.072 | nM | 8.97 |
| CHEMBL4863815 | — | IC50 | = | 1.107 | nM | 8.96 |
| CHEMBL4861227 | — | IC50 | = | 1.295 | nM | 8.89 |
| CHEMBL4863929 | — | IC50 | = | 1.348 | nM | 8.87 |