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Assay Detail

CHEMBL4880397

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
125I-labelled ET-1 saturation binding studies with EDNRA
1
Total Activities
1
Compounds Tested
1
Activity Types
1
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Endothelin-1 receptor (CHEMBL252)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Data for DCP probe A-192621
SGC Frankfurt
(2021)
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.25 5.25

Assay Parameters

Parameter Type Value Units Text
Assay publication Assay publication - PMID: 12193066

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL332794 A-192621 1 5.25

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL332794 A-192621 Ki = 5600.0 nM 5.25