Assay Detail
Binding
CHEMBL4882605
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NanoBRET (MAPK3, SGC Frankfurt)
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Data for DCP probe ERKi
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.17 | 5.17 |
| EC50 | 1 | 7.50 | 7.50 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4538174 | ERKi | — | 2 | 7.50 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4538174 | ERKi | EC50 | = | 32.0 | nM | 7.50 |
| CHEMBL4538174 | ERKi | IC50 | = | 6690.0 | nM | 5.17 |