Assay Detail
Binding
CHEMBL4883188
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Biochemical activity-MetAP2 using Mn
2
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Data for DCP probe TP-004
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 8.15 | 8.15 |
| Kd | 1 | 8.70 | 8.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4456585 | WM-1119 | — | 1 | 8.70 |
| CHEMBL3799512 | TP-004 | — | 1 | 8.15 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4456585 | WM-1119 | Kd | = | 2.0 | nM | 8.70 |
| CHEMBL3799512 | TP-004 | IC50 | = | 7.0 | nM | 8.15 |