Assay Detail
Binding
CHEMBL4883202
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NanoBRET (SGC Frankfurt) (CLK1)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Dual specificity protein kinase CLK1 (CHEMBL4224) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Data for DCP probe T3-CLK
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 8.46 | 8.46 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4531334 | T3-CLK | — | 1 | 8.46 |
| CHEMBL4576555 | T3-CLK-N | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4531334 | T3-CLK | IC50 | = | 3.49 | nM | 8.46 |
| CHEMBL4576555 | T3-CLK-N | IC50 | > | 10000.0 | nM | - |