Assay Detail
Binding
CHEMBL4884219
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AMPKalpha2(h) Eurofins kinase panel
2
Total Activities
1
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
5'-AMP-activated protein kinase catalytic subunit alpha-2 (CHEMBL2116) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Data for DCP probe BAY-3827
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| % residual kinase activity | 1 | - | - |
| IC50 | 1 | 8.15 | 8.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4580220 | BAY-3827 | — | 2 | 8.15 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4580220 | BAY-3827 | IC50 | = | 7.0 | nM | 8.15 |
| CHEMBL4580220 | BAY-3827 | % residual kinase activity | = | - | % | - |