Assay Detail
Binding
CHEMBL4884583
Review assay metadata, readout intent, target linkage, and publication context from the same page.
PRESTO-Tango concentration response assay
2
Total Activities
2
Compounds Tested
1
Activity Types
1
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Mas-related G-protein coupled receptor member X2 (CHEMBL5849) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Data for DCP probe (R)-ZINC-3573
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 6.13 | 6.13 |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| Assay publication | Assay publication | - | — | PMID: 28288109 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4520293 | (R)-ZINC-3573 | — | 1 | 6.13 |
| CHEMBL4534980 | (S)-ZINC-3573 | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4520293 | (R)-ZINC-3573 | EC50 | = | 740.0 | nM | 6.13 |
| CHEMBL4534980 | (S)-ZINC-3573 | EC50 | > | 100000.0 | nM | - |