Assay Detail

CHEMBL4884584

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Binding

FLIPR assay

ChEMBL ↗

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Target

Mas-related G-protein coupled receptor member X2 (CHEMBL5849) ↗

Open DB target context

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Mas-related G-protein coupled receptor member X2 (CHEMBL5849) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target Mas-related G-protein coupled receptor member X2

CHEMBL5849

Anchored from Assay target.

Protein identity Mas-related G-protein coupled receptor member X2

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Binding
Organism	Homo sapiens
Confidence	9 — Direct single protein target
Curated By	Autocuration

Target

Type	SINGLE PROTEIN
Organism	Homo sapiens

Publication

Data for DCP probe (R)-ZINC-3573

SGC Frankfurt
(2021)
· DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
EC50	2	6.00	6.00

Assay Parameters

Parameter	Type	Value	Units	Text
Assay publication	Assay publication	-	—	PMID: 28288109

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL4520293	(R)-ZINC-3573	—	1	6.00
CHEMBL4534980	(S)-ZINC-3573	—	1	-

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL4520293	(R)-ZINC-3573	EC50	=	1000.0	nM	6.00
CHEMBL4534980	(S)-ZINC-3573	EC50	>	100000.0	nM	-