Assay Detail
Binding
CHEMBL4884590
Review assay metadata, readout intent, target linkage, and publication context from the same page.
NanoBRET (SGC-Frankfurt) (DDR1)
2
Total Activities
2
Compounds Tested
1
Activity Types
2
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Epithelial discoidin domain-containing receptor 1 (CHEMBL5319) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Data for DCP probe SR-302
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.15 | 7.64 |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| Target protein length | Target protein length | - | — | full-length |
| Target protein type | Target protein type | - | — | HEK293T cells |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4591082 | SR-302 | — | 1 | 7.64 |
| CHEMBL4568183 | SR-301 | — | 1 | 4.66 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4591082 | SR-302 | IC50 | = | 23.0 | nM | 7.64 |
| CHEMBL4568183 | SR-301 | IC50 | = | 21900.0 | nM | 4.66 |