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Assay Detail

CHEMBL4886928

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding assay (LTB4R )
1
Total Activities
1
Compounds Tested
1
Activity Types
1
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Leukotriene B4 receptor 1 (CHEMBL3911)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Data for DCP probe PF-04418948
SGC Frankfurt
(2021)
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.32 5.32

Assay Parameters

Parameter Type Value Units Text
Assay publication Assay publication - PMID: 21595651

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3286797 PF-04418948 1.0 1 5.32

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3286797 PF-04418948 Ki = 4800.0 nM 5.32