Assay Detail
Binding
CHEMBL4887017
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ML2 (MT3) CEREP ligand profiling
3
Total Activities
1
Compounds Tested
3
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Ribosyldihydronicotinamide dehydrogenase [quinone] (CHEMBL3959) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Data for DCP probe PF-04418948
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Inhibition | 1 | - | - |
| IC50 | 1 | 6.28 | 6.28 |
| Ki | 1 | 6.28 | 6.28 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3286797 | PF-04418948 | 1.0 | 3 | 6.28 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3286797 | PF-04418948 | IC50 | = | 530.0 | nM | 6.28 |
| CHEMBL3286797 | PF-04418948 | Ki | = | 520.0 | nM | 6.28 |
| CHEMBL3286797 | PF-04418948 | Inhibition | = | 93.0 | % | - |