Assay Detail

CHEMBL4887159

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Binding

Dose response measurement (AAK1)

ChEMBL ↗

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Target

AP2-associated protein kinase 1 (CHEMBL3830) ↗

Open DB target context

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AP2-associated protein kinase 1 (CHEMBL3830) is the working anchor for this assay review. Loading the live Open DB target snapshot…

Primary target AP2-associated protein kinase 1

CHEMBL3830

Anchored from Assay target.

Protein identity AP2-associated protein kinase 1

Disease frame Disease evidence pending

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Review focus Open DB context pending

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Total Activities

Compounds Tested

Activity Types

Assay Parameters

Assay Information

Assay Type	Binding
Organism	Homo sapiens
Confidence	9 — Direct single protein target
Curated By	Autocuration

Target

AP2-associated protein kinase 1 (CHEMBL3830) ↗

Type	SINGLE PROTEIN
Organism	Homo sapiens

Publication

Data for DCP probe BI 605906

SGC Frankfurt
(2021)
· DOI

Activity Statistics

Type	Count	Avg pChEMBL	Best pChEMBL
IC50	1	6.57	6.57

Compounds Tested

Compound	Name	Phase	Activities	Best pChEMBL
CHEMBL4522930	BI-605906	—	1	6.57

Activity Data

Compound	Name	Type	Rel.	Value	Units	pChEMBL
CHEMBL4522930	BI-605906	IC50	=	272.0	nM	6.57