Assay Detail
Binding
CHEMBL4887759
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Eurofins Kinase panel (PIP4K2A)
2
Total Activities
2
Compounds Tested
1
Activity Types
1
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Phosphatidylinositol 5-phosphate 4-kinase type-2 alpha (CHEMBL1795194) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Data for DCP probe BAY-091
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.13 | 7.68 |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| Compound concentration | Compound concentration | 1.0 | uM | — |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4802045 | BAY-091 | — | 1 | 7.68 |
| CHEMBL4802048 | BAY-0361 | — | 1 | 6.57 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4802045 | BAY-091 | IC50 | = | 21.0 | nM | 7.68 |
| CHEMBL4802048 | BAY-0361 | IC50 | = | 271.0 | nM | 6.57 |