Assay Detail
Binding
CHEMBL5029258
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of jack bean alpha-mannosidase
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Canavalia ensiformis |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Positional Isomeric Effects on the Optical Properties, Multivalent Glycosidase Inhibition Effect, and Hypoglycemic Effect of Perylene Bisimide-deoxynojirimycin Conjugates.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 4 | 7.35 | 7.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5090920 | — | — | 1 | 7.77 |
| CHEMBL5078012 | — | — | 1 | 6.92 |
| CHEMBL1561 | MIGLITOL | 4.0 | 1 | - |
| CHEMBL5077606 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5090920 | — | Kd | = | 17.0 | nM | 7.77 |
| CHEMBL5078012 | — | Kd | = | 120.0 | nM | 6.92 |
| CHEMBL1561 | MIGLITOL | Kd | = | 105130.0 | nM | - |
| CHEMBL5077606 | — | Kd | = | 277320.0 | nM | - |