Assay Detail
Binding
CHEMBL5032883
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Induction of disruption of r(CCUG)12-MBNL1 complex (unknown origin) incubated for 15 mins by TR-FRET assay
82
Total Activities
82
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
A Druglike Small Molecule that Targets r(CCUG) Repeats in Myotonic Dystrophy Type 2 Facilitates Degradation by RNA Quality Control Pathways.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 82 | 4.63 | 6.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5087124 | — | — | 1 | 6.70 |
| CHEMBL5078834 | — | — | 1 | 6.52 |
| CHEMBL5089176 | — | — | 1 | 6.52 |
| CHEMBL5092071 | — | — | 1 | 6.40 |
| CHEMBL5075325 | — | — | 1 | 6.00 |
| CHEMBL5079565 | — | — | 1 | 6.00 |
| CHEMBL5085783 | — | — | 1 | 5.70 |
| CHEMBL5090835 | — | — | 1 | 5.40 |
| CHEMBL5093033 | — | — | 1 | 5.16 |
| CHEMBL5079182 | — | — | 1 | 5.00 |
| CHEMBL5086011 | — | — | 1 | 5.00 |
| CHEMBL5085100 | — | — | 1 | 5.00 |
| CHEMBL5087841 | — | — | 1 | 5.00 |
| CHEMBL5094054 | — | — | 1 | 4.82 |
| CHEMBL5088202 | — | — | 1 | 4.70 |
| CHEMBL5083599 | — | — | 1 | 4.70 |
| CHEMBL5078110 | — | — | 1 | 4.52 |
| CHEMBL5088264 | — | — | 1 | 4.52 |
| CHEMBL5085754 | — | — | 1 | 4.52 |
| CHEMBL5077669 | — | — | 1 | 4.46 |
| CHEMBL3808617 | — | — | 1 | 4.40 |
| CHEMBL5094908 | — | — | 1 | 4.40 |
| CHEMBL4082535 | — | — | 1 | 4.35 |
| CHEMBL5086427 | — | — | 1 | 4.30 |
| CHEMBL5083630 | — | — | 1 | 4.30 |
| CHEMBL5070611 | — | — | 1 | 4.30 |
| CHEMBL5092427 | — | — | 1 | 4.22 |
| CHEMBL5080960 | — | — | 1 | 4.22 |
| CHEMBL5087804 | — | — | 1 | 4.22 |
| CHEMBL5093361 | — | — | 1 | 4.19 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5087124 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL5078834 | — | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL5089176 | — | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL5092071 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL5075325 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL5079565 | — | IC50 | = | 1000.0 | nM | 6.00 |
| CHEMBL5085783 | — | IC50 | = | 2000.0 | nM | 5.70 |
| CHEMBL5090835 | — | IC50 | = | 4000.0 | nM | 5.40 |
| CHEMBL5093033 | — | IC50 | = | 7000.0 | nM | 5.16 |
| CHEMBL5079182 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL5086011 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL5085100 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL5087841 | — | IC50 | = | 10000.0 | nM | 5.00 |
| CHEMBL5094054 | — | IC50 | = | 15000.0 | nM | 4.82 |
| CHEMBL5083599 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL5088202 | — | IC50 | = | 20000.0 | nM | 4.70 |
| CHEMBL5078110 | — | IC50 | = | 30000.0 | nM | 4.52 |
| CHEMBL5088264 | — | IC50 | = | 30000.0 | nM | 4.52 |
| CHEMBL5085754 | — | IC50 | = | 30000.0 | nM | 4.52 |
| CHEMBL5077669 | — | IC50 | = | 35000.0 | nM | 4.46 |
| CHEMBL3808617 | — | IC50 | = | 40000.0 | nM | 4.40 |
| CHEMBL5094908 | — | IC50 | = | 40000.0 | nM | 4.40 |
| CHEMBL4082535 | — | IC50 | = | 45000.0 | nM | 4.35 |
| CHEMBL5070611 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL5086427 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL5083630 | — | IC50 | = | 50000.0 | nM | 4.30 |
| CHEMBL5092427 | — | IC50 | = | 60000.0 | nM | 4.22 |
| CHEMBL5080960 | — | IC50 | = | 60000.0 | nM | 4.22 |
| CHEMBL5087804 | — | IC50 | = | 60000.0 | nM | 4.22 |
| CHEMBL5093361 | — | IC50 | = | 65000.0 | nM | 4.19 |
| CHEMBL5094335 | — | IC50 | = | 70000.0 | nM | 4.16 |
| CHEMBL5083215 | — | IC50 | = | 70000.0 | nM | 4.16 |
| CHEMBL5087066 | — | IC50 | = | 70000.0 | nM | 4.16 |
| CHEMBL5077362 | — | IC50 | = | 70000.0 | nM | 4.16 |
| CHEMBL5076423 | — | IC50 | = | 70000.0 | nM | 4.16 |
| CHEMBL5088344 | — | IC50 | = | 70000.0 | nM | 4.16 |
| CHEMBL5093070 | — | IC50 | = | 75000.0 | nM | 4.12 |
| CHEMBL5092670 | — | IC50 | = | 75000.0 | nM | 4.12 |
| CHEMBL5075311 | — | IC50 | = | 80000.0 | nM | 4.10 |
| CHEMBL5089460 | — | IC50 | = | 80000.0 | nM | 4.10 |
| CHEMBL527587 | — | IC50 | = | 80000.0 | nM | 4.10 |
| CHEMBL5094946 | — | IC50 | = | 85000.0 | nM | 4.07 |
| CHEMBL5093819 | — | IC50 | = | 85000.0 | nM | 4.07 |
| CHEMBL5094434 | — | IC50 | = | 90000.0 | nM | 4.05 |
| CHEMBL5083698 | — | IC50 | = | 90000.0 | nM | 4.05 |
| CHEMBL5094375 | — | IC50 | = | 95000.0 | nM | 4.02 |
| CHEMBL5079615 | — | IC50 | = | 95000.0 | nM | 4.02 |
| CHEMBL5079447 | — | IC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL5087836 | — | IC50 | = | 100000.0 | nM | 4.00 |
| CHEMBL5079164 | — | IC50 | = | 100000.0 | nM | 4.00 |