Assay Detail
Binding
CHEMBL5037539
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Displacement of kinase tracer 236 from TTK (unknown origin) by LanthaScreen Eu kinase binding assay
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Structure-Guided Optimization Provides a Series of TTK Protein Inhibitors with Potent Antitumor Activity.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 17 | 8.51 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5093015 | — | — | 1 | 9.00 |
| CHEMBL5092826 | — | — | 1 | 9.00 |
| CHEMBL5081270 | — | — | 1 | 8.70 |
| CHEMBL5075313 | — | — | 1 | 8.70 |
| CHEMBL5073101 | — | — | 1 | 8.70 |
| CHEMBL5077668 | — | — | 1 | 8.70 |
| CHEMBL5081668 | — | — | 1 | 8.55 |
| CHEMBL5084062 | — | — | 1 | 8.52 |
| CHEMBL5091689 | — | — | 1 | 8.52 |
| CHEMBL5085753 | — | — | 1 | 8.52 |
| CHEMBL5085278 | — | — | 1 | 8.40 |
| CHEMBL5086022 | — | — | 1 | 8.40 |
| CHEMBL5079606 | — | — | 1 | 8.28 |
| CHEMBL5085182 | — | — | 1 | 8.25 |
| CHEMBL5086435 | — | — | 1 | 8.22 |
| CHEMBL5077627 | — | — | 1 | 8.12 |
| CHEMBL5087340 | — | — | 1 | 8.05 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5093015 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL5092826 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL5081270 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL5075313 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL5073101 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL5077668 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL5081668 | — | IC50 | = | 2.8 | nM | 8.55 |
| CHEMBL5084062 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL5091689 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL5085753 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL5085278 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL5086022 | — | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL5079606 | — | IC50 | = | 5.3 | nM | 8.28 |
| CHEMBL5085182 | — | IC50 | = | 5.6 | nM | 8.25 |
| CHEMBL5086435 | — | IC50 | = | 6.0 | nM | 8.22 |
| CHEMBL5077627 | — | IC50 | = | 7.5 | nM | 8.12 |
| CHEMBL5087340 | — | IC50 | = | 9.0 | nM | 8.05 |