Assay Detail
Functional
CHEMBL5058654
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Eurofins cellular functional assay - Antagonist (EDNRA)
3
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Data for DCP probe A-192621
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 5.68 | 5.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4533479 | A-1806262 | — | 2 | 5.80 |
| CHEMBL332794 | A-192621 | — | 1 | 5.44 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4533479 | A-1806262 | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL4533479 | A-1806262 | IC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL332794 | A-192621 | IC50 | = | 3600.0 | nM | 5.44 |