Assay Detail
Binding
CHEMBL5096567
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Inhibition of NUAK1 (unknown origin)
14
Total Activities
14
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Development and Therapeutic Potential of NUAKs Inhibitors.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 14 | 7.54 | 8.85 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5176650 | — | — | 1 | 8.85 |
| CHEMBL5199998 | — | — | 1 | 8.52 |
| CHEMBL4116008 | CERDULATINIB | 2.0 | 1 | 8.40 |
| CHEMBL5196626 | — | — | 1 | 8.32 |
| CHEMBL577784 | BX-795 | — | 1 | 8.30 |
| CHEMBL5204647 | — | — | 1 | 8.04 |
| CHEMBL5169640 | — | — | 1 | 7.46 |
| CHEMBL3545311 | BRIGATINIB | 4.0 | 1 | 7.33 |
| CHEMBL535 | SUNITINIB | 4.0 | 1 | 7.32 |
| CHEMBL3544911 | PREXASERTIB | 2.0 | 1 | 7.19 |
| CHEMBL3605057 | — | — | 1 | 6.64 |
| CHEMBL5182271 | — | — | 1 | 6.39 |
| CHEMBL5200931 | — | — | 1 | 5.30 |
| CHEMBL4442620 | RONICICLIB | 2.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5176650 | — | IC50 | = | 1.4 | nM | 8.85 |
| CHEMBL5199998 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL4116008 | CERDULATINIB | IC50 | = | 4.0 | nM | 8.40 |
| CHEMBL5196626 | — | IC50 | = | 4.8 | nM | 8.32 |
| CHEMBL577784 | BX-795 | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL5204647 | — | IC50 | = | 9.1 | nM | 8.04 |
| CHEMBL5169640 | — | IC50 | = | 34.9 | nM | 7.46 |
| CHEMBL3545311 | BRIGATINIB | IC50 | = | 47.0 | nM | 7.33 |
| CHEMBL535 | SUNITINIB | IC50 | = | 48.0 | nM | 7.32 |
| CHEMBL3544911 | PREXASERTIB | IC50 | = | 64.0 | nM | 7.19 |
| CHEMBL3605057 | — | IC50 | = | 230.0 | nM | 6.64 |
| CHEMBL5182271 | — | IC50 | = | 411.0 | nM | 6.39 |
| CHEMBL5200931 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL4442620 | RONICICLIB | IC50 | < | 10.0 | nM | - |