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Assay Detail

CHEMBL5096644

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity to human GPR55 expressed in HEK293 cells assessed as LPI-stimulated ERK1/2 phosphorylation
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type HEK293
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

G-protein coupled receptor 55 (CHEMBL1075322)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Phytocannabinoid Pharmacology: Medicinal Properties of <i>Cannabis sativa</i> Constituents Aside from the "Big Two".
Sampson PB.
J Nat Prod (2021) 84 : 142 -160
PubMed 33356248 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 6.40 6.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2387742 CANNABIDIVARIN 2.0 1 6.40

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2387742 CANNABIDIVARIN EC50 = 400.0 nM 6.40