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Assay Detail

CHEMBL5096672

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Displacement of [3H]-WIN55212-2 from human CB2 receptor transfected in CHO cell membrane incubated for 90 mins by Liquid scintillation counter analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Cell Type CHO
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Cannabinoid receptor 2 (CHEMBL253)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Phytocannabinoid Pharmacology: Medicinal Properties of <i>Cannabis sativa</i> Constituents Aside from the "Big Two".
Sampson PB.
J Nat Prod (2021) 84 : 142 -160
PubMed 33356248 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.91 5.91

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL497318 CANNABIGEROL 2.0 1 5.91

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL497318 CANNABIGEROL Ki = 1220.0 nM 5.91