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Assay Detail

CHEMBL5098050

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of recombinant His-tagged wild-type HIV-1 group M subtype B BH10 reverse transcriptase-associated RNase H activity harboring p66/p51 hetrodimer expressed in Escherichia coli M15 using GTTTTCTTTTCCCCCCTGAC-30 fluorescein/50-CAAAAGAAAAGGGGGGACUG-30 Dabcyl RNA/DNA template-primer as substrate incubated for 1 hr by multilabel counter plate reader analysis
40
Total Activities
40
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Human immunodeficiency virus 1
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Human immunodeficiency virus type 1 reverse transcriptase (CHEMBL247)
Type SINGLE PROTEIN
Organism Human immunodeficiency virus 1

Publication

Quinolinonyl Non-Diketo Acid Derivatives as Inhibitors of HIV-1 Ribonuclease H and Polymerase Functions of Reverse Transcriptase.
Messore A, Corona A, Madia VN, Saccoliti F, Tudino V, De Leo A, Ialongo D, Scipione L, De Vita D, Amendola G, Novellino E, Cosconati S, Métifiot M, Andreola ML, Esposito F, Grandi N, Tramontano E, Costi R, Di Santo R.
J Med Chem (2021) 64 : 8579 -8598
PubMed 34106711 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 40 4.80 6.72

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL550937 BETA-THUJAPLICINOL 1 6.72
CHEMBL5172754 1 5.83
CHEMBL5173288 1 5.82
CHEMBL5176128 1 5.23
CHEMBL5198310 1 5.13
CHEMBL5185855 1 5.13
CHEMBL5174596 1 5.10
CHEMBL5197780 1 5.09
CHEMBL5202973 1 5.08
CHEMBL5194402 1 4.96
CHEMBL5183730 1 4.87
CHEMBL5187082 1 4.82
CHEMBL5187446 1 4.81
CHEMBL5207303 1 4.79
CHEMBL5191482 1 4.71
CHEMBL5182942 1 4.62
CHEMBL5184868 1 4.55
CHEMBL5198940 1 4.53
CHEMBL5172266 1 4.52
CHEMBL5171239 1 4.50
CHEMBL5188823 1 4.47
CHEMBL5191403 1 4.43
CHEMBL5192134 1 4.34
CHEMBL5175570 1 4.32
CHEMBL5179284 1 4.26
CHEMBL3309770 1 4.25
CHEMBL5201776 1 4.23
CHEMBL5185881 1 4.13
CHEMBL5172028 1 4.00
CHEMBL5208591 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL550937 BETA-THUJAPLICINOL IC50 = 190.0 nM 6.72
CHEMBL5172754 IC50 = 1490.0 nM 5.83
CHEMBL5173288 IC50 = 1510.0 nM 5.82
CHEMBL5176128 IC50 = 5900.0 nM 5.23
CHEMBL5198310 IC50 = 7470.0 nM 5.13
CHEMBL5185855 IC50 = 7480.0 nM 5.13
CHEMBL5174596 IC50 = 8000.0 nM 5.10
CHEMBL5197780 IC50 = 8190.0 nM 5.09
CHEMBL5202973 IC50 = 8270.0 nM 5.08
CHEMBL5194402 IC50 = 11000.0 nM 4.96
CHEMBL5183730 IC50 = 13500.0 nM 4.87
CHEMBL5187082 IC50 = 15300.0 nM 4.82
CHEMBL5187446 IC50 = 15400.0 nM 4.81
CHEMBL5207303 IC50 = 16300.0 nM 4.79
CHEMBL5191482 IC50 = 19600.0 nM 4.71
CHEMBL5182942 IC50 = 24000.0 nM 4.62
CHEMBL5184868 IC50 = 28400.0 nM 4.55
CHEMBL5198940 IC50 = 29500.0 nM 4.53
CHEMBL5172266 IC50 = 30300.0 nM 4.52
CHEMBL5171239 IC50 = 32000.0 nM 4.50
CHEMBL5188823 IC50 = 34000.0 nM 4.47
CHEMBL5191403 IC50 = 37200.0 nM 4.43
CHEMBL5192134 IC50 = 45500.0 nM 4.34
CHEMBL5175570 IC50 = 47800.0 nM 4.32
CHEMBL5179284 IC50 = 55300.0 nM 4.26
CHEMBL3309770 IC50 = 56000.0 nM 4.25
CHEMBL5201776 IC50 = 59000.0 nM 4.23
CHEMBL5185881 IC50 = 74000.0 nM 4.13
CHEMBL5172028 IC50 = 100000.0 nM 4.00
CHEMBL5173434 IC50 > 100000.0 nM -
CHEMBL5180442 IC50 > 100000.0 nM -
CHEMBL5171586 IC50 > 100000.0 nM -
CHEMBL4648347 IC50 > 100000.0 nM -
CHEMBL5205380 IC50 > 100000.0 nM -
CHEMBL5188713 IC50 > 100000.0 nM -
CHEMBL5208821 IC50 > 100000.0 nM -
CHEMBL5182985 IC50 > 100000.0 nM -
CHEMBL5183793 IC50 > 100000.0 nM -
CHEMBL5193857 IC50 > 100000.0 nM -
CHEMBL5208591 IC50 > 100000.0 nM -