Assay Detail
Functional
CHEMBL5108116
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human CB2R expressed in mouse AtT20 cells by FLIPR membrane potential assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | AtT20 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Synthesis and antitumour evaluation of indole-2-carboxamides against paediatric brain cancer cells.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 7.21 | 7.21 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1592888 | — | — | 1 | 7.21 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1592888 | — | EC50 | = | 62.0 | nM | 7.21 |