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Assay Detail

CHEMBL5127935

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Functional
Antiproliferative activity against human HAL-01 cells assessed as cell growth inhibition by MTT assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HAL-01
Confidence 1 — Organism
Curated By Autocuration

Target

HAL-01 (CHEMBL2366142)
Type CELL-LINE
Organism Homo sapiens

Publication

Drug discovery of histone lysine demethylases (KDMs) inhibitors (progress from 2018 to present).
He X, Zhang H, Zhang Y, Ye Y, Wang S, Bai R, Xie T, Ye XY.
Eur J Med Chem (2022) 231 : 114143 -114143
PubMed 35101649 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.96 5.96

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5201233 1 5.96

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5201233 IC50 = 1100.0 nM 5.96