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Assay Detail

CHEMBL5128286

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against Ebola virus pseudotyped infected in HEK293T cells assessed as reduction in viral cytopathic effect
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Ebolavirus
Cell Type HEK-293T
Confidence 1 — Organism
Curated By Autocuration

Target

Ebolavirus (CHEMBL4434621)
Type ORGANISM
Organism Ebolavirus

Publication

Recent applications of vinyl sulfone motif in drug design and discovery.
Ahmadi R, Emami S.
Eur J Med Chem (2022) 234 : 114255 -114255
PubMed 35305462 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 10.26 10.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5190923 1 10.40
CHEMBL5185113 1 10.40
CHEMBL5181012 1 10.40
CHEMBL5198546 1 10.40
CHEMBL4743491 1 10.40
CHEMBL4755358 1 10.40
CHEMBL91704 K-777 2.0 1 9.44

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5190923 IC50 = 0.04 nM 10.40
CHEMBL5185113 IC50 = 0.04 nM 10.40
CHEMBL5181012 IC50 = 0.04 nM 10.40
CHEMBL5198546 IC50 = 0.04 nM 10.40
CHEMBL4743491 IC50 = 0.04 nM 10.40
CHEMBL4755358 IC50 = 0.04 nM 10.40
CHEMBL91704 K-777 IC50 = 0.36 nM 9.44