Assay Detail
Binding
CHEMBL5131963
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Binding affinity to AAK1 (unknown origin) assessed as dissociation constant
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Kinase Inhibitors as Underexplored Antiviral Agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 11 | 7.96 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5200929 | — | — | 1 | 9.00 |
| CHEMBL5184366 | — | — | 1 | 9.00 |
| CHEMBL4439128 | — | — | 1 | 8.40 |
| CHEMBL2105759 | BARICITINIB | 4.0 | 1 | 8.09 |
| CHEMBL4452939 | — | — | 1 | 8.04 |
| CHEMBL535 | SUNITINIB | 4.0 | 1 | 7.96 |
| CHEMBL516312 | — | — | 1 | 7.28 |
| CHEMBL553 | ERLOTINIB | 4.0 | 1 | 5.92 |
| CHEMBL4458078 | — | — | 1 | - |
| CHEMBL5416410 | DASATINIB | 4.0 | 1 | - |
| CHEMBL939 | GEFITINIB | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5200929 | — | Kd | = | 1.0 | nM | 9.00 |
| CHEMBL5184366 | — | Kd | = | 1.0 | nM | 9.00 |
| CHEMBL4439128 | — | Kd | = | 4.0 | nM | 8.40 |
| CHEMBL2105759 | BARICITINIB | Kd | = | 8.2 | nM | 8.09 |
| CHEMBL4452939 | — | Kd | = | 9.1 | nM | 8.04 |
| CHEMBL535 | SUNITINIB | Kd | = | 11.0 | nM | 7.96 |
| CHEMBL516312 | — | Kd | = | 53.0 | nM | 7.28 |
| CHEMBL553 | ERLOTINIB | Kd | = | 1200.0 | nM | 5.92 |
| CHEMBL4458078 | — | Kd | = | 18000000.0 | nM | - |
| CHEMBL5416410 | DASATINIB | Kd | > | 3000.0 | nM | - |
| CHEMBL939 | GEFITINIB | Kd | > | 3000.0 | nM | - |