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Assay Detail

CHEMBL5140840

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Potentiation of vancomycin-induced antibacterial activity against methicillin resistant Staphylococcus aureus Mu50 in presence of vancomycin
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Staphylococcus aureus
Confidence 1 — Organism
Curated By Autocuration

Target

Staphylococcus aureus (CHEMBL352)
Type ORGANISM
Organism Staphylococcus aureus

Publication

Small Carbohydrate Derivatives as Potent Antibiofilm Agents.
Singh K, Kulkarni SS.
J Med Chem (2022) 65 : 8525 -8549
PubMed 35777073 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 6 5.32 5.90

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4078565 1 5.90
CHEMBL4072752 1 5.43
CHEMBL4077423 1 5.10
CHEMBL3590184 1 5.10
CHEMBL5205021 1 5.08
CHEMBL491592 HAMAMELITANNIN 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4078565 EC50 = 1270.0 nM 5.90
CHEMBL4072752 EC50 = 3710.0 nM 5.43
CHEMBL4077423 EC50 = 7980.0 nM 5.10
CHEMBL3590184 EC50 = 7970.0 nM 5.10
CHEMBL5205021 EC50 = 8290.0 nM 5.08
CHEMBL491592 HAMAMELITANNIN EC50 = 165000.0 nM -