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Assay Detail

CHEMBL5140879

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Pseudomonas aeruginosa LecB incubated for 8 to 22 hrs by fluorescence polarization based competitive binding analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Pseudomonas aeruginosa
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Fucose-binding lectin PA-IIL (CHEMBL4523938)
Type SINGLE PROTEIN
Organism Pseudomonas aeruginosa (strain ATCC 15692 / DSM 22644 / CIP 104116 / JCM14847 / LMG 12228 / 1C / PRS 101 / PAO1)

Publication

Small Carbohydrate Derivatives as Potent Antibiofilm Agents.
Singh K, Kulkarni SS.
J Med Chem (2022) 65 : 8525 -8549
PubMed 35777073 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 4.67 4.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4450053 1 4.70
CHEMBL3800313 1 4.64

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4450053 IC50 = 20000.0 nM 4.70
CHEMBL3800313 IC50 = 23000.0 nM 4.64