Assay Detail
Binding
CHEMBL5140919
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]mibolerone from Androgen receptor (unknown origin) measured by liquid scintillation counting method
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Therapeutic Strategies to Target the Androgen Receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 8.83 | 9.26 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1738889 | ENOBOSARM | 3.0 | 1 | 9.26 |
| CHEMBL125236 | — | — | 1 | 8.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1738889 | ENOBOSARM | Ki | = | 0.55 | nM | 9.26 |
| CHEMBL125236 | — | Ki | = | 4.0 | nM | 8.40 |