Assay Detail
Binding
CHEMBL5140920
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at Androgen receptor (unknown origin)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Therapeutic Strategies to Target the Androgen Receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 8.54 | 8.74 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL229861 | — | — | 1 | 8.74 |
| CHEMBL4088914 | — | — | 1 | 8.33 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL229861 | — | EC50 | = | 1.8 | nM | 8.74 |
| CHEMBL4088914 | — | EC50 | = | 4.7 | nM | 8.33 |