Assay Detail
Binding
CHEMBL5140925
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at Androgen receptor (unknown origin) transfected in mouse C2C12 cells measured by luciferase reporter assay
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Cell Type | C2C12 |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Therapeutic Strategies to Target the Androgen Receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 8.62 | 9.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3326454 | — | — | 1 | 9.30 |
| CHEMBL229264 | — | — | 1 | 8.64 |
| CHEMBL233773 | — | — | 1 | 7.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3326454 | — | EC50 | = | 0.5 | nM | 9.30 |
| CHEMBL229264 | — | EC50 | = | 2.3 | nM | 8.64 |
| CHEMBL233773 | — | EC50 | = | 11.9 | nM | 7.92 |