Assay Detail
Binding
CHEMBL5140955
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at human Androgen receptor measured by AR-mediated transcriptional activation assay
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Therapeutic Strategies to Target the Androgen Receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.83 | 6.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL197595 | — | — | 1 | 6.96 |
| CHEMBL202990 | — | — | 1 | 6.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL197595 | — | IC50 | = | 110.0 | nM | 6.96 |
| CHEMBL202990 | — | IC50 | = | 200.0 | nM | 6.70 |