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Assay Detail

CHEMBL5140958

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiproliferative activity against human LNCaP cells expressing wild-type Androgen receptor
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type LNCaP
Confidence 1 — Organism
Curated By Autocuration

Target

LNCaP (CHEMBL612518)
Type CELL-LINE
Organism Homo sapiens

Publication

Therapeutic Strategies to Target the Androgen Receptor.
Xiang W, Wang S.
J Med Chem (2022) 65 : 8772 -8797
PubMed 35786895 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 6.54 6.54

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL2337513 1 6.54

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL2337513 IC50 = 290.0 nM 6.54