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Assay Detail

CHEMBL5146630

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Toxicity
Cytotoxicity against human HaCaT cells assessed as reduction in cell viability incubated for 24 hrs by CellTiter-Blue cell viability assay
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Toxicity
Organism Homo sapiens
Cell Type HaCaT
Confidence 1 — Organism
Curated By Autocuration

Target

HaCaT (CHEMBL614392)
Type CELL-LINE
Organism Homo sapiens

Publication

Antimicrobial Prenylated Isoflavones from the Leaves of the Amazonian Medicinal Plant <i>Vatairea guianensis</i> Aubl.
Çiçek SS, Galarza Pérez M, Wenzel-Storjohann A, Bezerra RM, Segovia JFO, Girreser U, Kanzaki I, Tasdemir D.
J Nat Prod (2022) 85 : 927 -935
PubMed 35271771 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 4.16 4.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL53463 DOXORUBICIN 4.0 1 4.30
CHEMBL5174986 1 4.16
CHEMBL5170827 1 4.09
CHEMBL5177554 1 4.07
CHEMBL3616491 1 -
CHEMBL5172980 1 -
CHEMBL5180194 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL53463 DOXORUBICIN IC50 = 50000.0 nM 4.30
CHEMBL5174986 IC50 = 69800.0 nM 4.16
CHEMBL5170827 IC50 = 80700.0 nM 4.09
CHEMBL5177554 IC50 = 85900.0 nM 4.07
CHEMBL3616491 IC50 = 159800.0 nM -
CHEMBL5172980 IC50 = 134600.0 nM -
CHEMBL5180194 IC50 = 207000.0 nM -